Cargando...

Late-Stage Diversification of Biologically Active Molecules via Chemoenzymatic C-H Functionalization

Engineered variants of rebeccamycin halogenase were used to selectively halogenate a number of biologically active aromatic compounds. Subsequent Pd-catalyzed cross-coupling reactions on the crude extracts of these reactions were used to install aryl, amine, and ether substituents at the halogenatio...

Descrición completa

Gardado en:
Detalles Bibliográficos
Publicado en:ACS Catal
Main Authors: Durak, Landon J., Payne, James T., Lewis, Jared C.
Formato: Artigo
Idioma:Inglês
Publicado: 2016
Assuntos:
Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC4890977/
https://ncbi.nlm.nih.gov/pubmed/27274902
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acscatal.5b02558
Tags: Engadir etiqueta
Sen Etiquetas, Sexa o primeiro en etiquetar este rexistro!