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Sodium channel slow inactivation interferes with open channel block

Mutations in the voltage-gated sodium channel Nav1.7 are linked to inherited pain syndromes such as erythromelalgia (IEM) and paroxysmal extreme pain disorder (PEPD). PEPD mutations impair Nav1.7 fast inactivation and increase persistent currents. PEPD mutations also increase resurgent currents, whi...

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Publicat a:Sci Rep
Autors principals: Hampl, Martin, Eberhardt, Esther, O’Reilly, Andrias O., Lampert, Angelika
Format: Artigo
Idioma:Inglês
Publicat: Nature Publishing Group 2016
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4865801/
https://ncbi.nlm.nih.gov/pubmed/27174182
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/srep25974
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