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Distinct Pharmacodynamic Activity of Rilpivirine in Ectocervical and Colonic Explant Tissue

A long-acting injectable form of rilpivirine (RPV) is being evaluated in clinical trials for the prevention of HIV infection. Preclinical testing was undertaken to define RPV pharmacokinetic (PK) and pharmacodynamic (PD) activities in ectocervical and colonic tissue treated in vitro. Tenfold dilutio...

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Detalhes bibliográficos
Publicado no:Antimicrob Agents Chemother
Main Authors: Dezzutti, Charlene S., Else, Laura J., Yandura, Sarah E., Shetler, Cory, Russo, Julie, Back, David J., McGowan, Ian
Formato: Artigo
Idioma:Inglês
Publicado em: American Society for Microbiology 2016
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4862523/
https://ncbi.nlm.nih.gov/pubmed/26902757
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.00167-16
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