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In vitro and in vivo drug disposition of cilengitide in animals and human

Cilengitide is very low permeable (1.0 nm/sec) stable cyclic pentapeptide containing an Arg‐Gly‐Asp motif responsible for selective binding to αvβ3 and αvβ5 integrins administered intravenously (i.v.). In vivo studies in the mouse and Cynomolgus monkeys showed the major component in plasma was uncha...

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Detalhes bibliográficos
Publicado no:Pharmacol Res Perspect
Main Authors: Dolgos, Hugues, Freisleben, Achim, Wimmer, Elmar, Scheible, Holger, Krätzer, Friedrich, Yamagata, Tetsuo, Gallemann, Dieter, Fluck, Markus
Formato: Artigo
Idioma:Inglês
Publicado em: John Wiley and Sons Inc. 2016
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4804314/
https://ncbi.nlm.nih.gov/pubmed/27069630
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/prp2.217
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