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Eukaryotic elongation factor 2 kinase as a drug target in cancer, and in cardiovascular and neurodegenerative diseases

Eukaryotic elongation factor 2 kinase (eEF2K) is an unusual protein kinase that regulates the elongation stage of protein synthesis by phosphorylating and inhibiting its only known substrate, eEF2. Elongation is a highly energy-consuming process, and eEF2K activity is tightly regulated by several si...

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Publicat a:Acta Pharmacol Sin
Autors principals: Liu, Rui, Proud, Christopher G
Format: Artigo
Idioma:Inglês
Publicat: Nature Publishing Group 2016
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4775846/
https://ncbi.nlm.nih.gov/pubmed/26806303
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/aps.2015.123
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