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Thermodynamics and kinetics of amphotericin B self-association in aqueous solution characterized in molecular detail

Amphotericin B (AmB) is a potent but toxic drug commonly used to treat systemic mycoses. Its efficiency as a therapeutic agent depends on its ability to discriminate between mammalian and fungal cell membranes. The association of AmB monomers in an aqueous environment plays an important role in drug...

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Detalhes bibliográficos
Publicado no:Sci Rep
Main Authors: Zielińska, Joanna, Wieczór, Miłosz, Bączek, Tomasz, Gruszecki, Marcin, Czub, Jacek
Formato: Artigo
Idioma:Inglês
Publicado em: Nature Publishing Group 2016
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4705489/
https://ncbi.nlm.nih.gov/pubmed/26742886
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/srep19109
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