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CYP2C8 Is a Novel Target of Peroxisome Proliferator-Activated Receptor α in Human Liver

Human cytochrome P450 (CYP) 2C enzymes metabolize ∼30% of clinically prescribed drugs and various environmental chemicals. CYP2C8, an important member of this subfamily, metabolizes the anticancer drug paclitaxel, certain antidiabetic drugs, and endogenous substrates, including arachidonic acid, to...

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Publicat a:Mol Pharmacol
Autors principals: Makia, Ngome L., Goldstein, Joyce A.
Format: Artigo
Idioma:Inglês
Publicat: The American Society for Pharmacology and Experimental Therapeutics 2016
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4702104/
https://ncbi.nlm.nih.gov/pubmed/26467040
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.115.100255
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