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pH-dependent population shift regulates BACE1 activity and inhibition

BACE1, a major therapeutic target for treatment of Alzheimer’s disease, functions within a narrow pH range. Despite tremendous effort and progress in the development of BACE1 inhibitors, details of the underlying pH-dependent regulatory mechanism remain unclear. Here we elucidate the pH-dependent co...

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Dettagli Bibliografici
Pubblicato in:J Am Chem Soc
Autori principali: Ellis, Christopher R., Shen, Jana
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2015
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4697946/
https://ncbi.nlm.nih.gov/pubmed/26186663
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jacs.5b05891
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