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An Umpolung Strategy for the Synthesis of β-Aminoketones via Copper-Catalyzed Electrophilic Amination of Cyclopropanols

A novel copper-catalyzed electrophilic amination of cyclopropanols with O-benzoyl-N,-N-dialkylhydroxylamines to synthesize various β-aminoketones via a sequence of C-C bond cleavage and C(sp3)-N bond formation is reported. The reaction conditions are mild and tolerate a wide range of functional grou...

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Bibliographic Details
Published in:Org Lett
Main Authors: Ye, Zhishi, Dai, Mingji
Format: Artigo
Language:Inglês
Published: 2015
Subjects:
Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC4690534/
https://ncbi.nlm.nih.gov/pubmed/25885943
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.orglett.5b00828
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