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Metal-Free, Efficient Hydrazination of Imidazo[1,2-a]pyridine with Diethyl Azodicarboxylate in Neutral Media

The first example of metal-free regioselective hydrazination of imidazo[1,2-a]pyridine with diethyl azodicarboxylate was accomplished. This procedure is chemically appealing due to the high degree of functional group tolerance and efficiency in expanding molecule diversity.

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Dades bibliogràfiques
Publicat a:Org Biomol Chem
Autors principals: Wang, Yuanxiang, Frett, Brendan, McConnell, Nick, Li, Hong-yu
Format: Artigo
Idioma:Inglês
Publicat: 2015
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4675458/
https://ncbi.nlm.nih.gov/pubmed/25611884
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c4ob02284j
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