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Selective Phosphodiesterase Inhibitors for Psoriasis: Focus on Apremilast

Phosphodiesterase (PDE) 4 participates in regulating the inflammatory response by degrading cyclic adenosine 3′,5′-monophosphate (cAMP), a key second messenger. Inhibition of PDE4 increases the intracellular cAMP level, which in turn results in a reduction in inflammatory mediators and an increase i...

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Foilsithe in:BioDrugs
Main Authors: Gooderham, Melinda, Papp, Kim
Formáid: Artigo
Teanga:Inglês
Foilsithe: Springer International Publishing 2015
Ábhair:
Rochtain Ar Líne:https://ncbi.nlm.nih.gov/pmc/articles/PMC4626529/
https://ncbi.nlm.nih.gov/pubmed/26481941
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s40259-015-0144-3
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