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Physiologically-based Pharmacokinetic Modeling of Target-Mediated Drug Disposition of Bortezomib in Mice

Bortezomib is a reversible proteasome inhibitor with potent antineoplastic activity that exhibits dose- and time-dependent pharmacokinetics (PK). Proteasome-mediated bortezomib disposition is proposed as the primary source of its nonlinear and apparent nonstationary PK behavior. Single intravenous (...

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Pubblicato in:J Pharmacokinet Pharmacodyn
Autori principali: Zhang, Li, Mager, Donald E.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2015
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4620045/
https://ncbi.nlm.nih.gov/pubmed/26391023
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s10928-015-9445-x
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