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Mutation of Rv2887, a marR-Like Gene, Confers Mycobacterium tuberculosis Resistance to an Imidazopyridine-Based Agent

Drug resistance is a major problem in Mycobacterium tuberculosis control, and it is critical to identify novel drug targets and new antimycobacterial compounds. We have previously identified an imidazo[1,2-a]pyridine-4-carbonitrile-based agent, MP-III-71, with strong activity against M. tuberculosis...

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Detalhes bibliográficos
Publicado no:Antimicrob Agents Chemother
Main Authors: Winglee, Kathryn, Lun, Shichun, Pieroni, Marco, Kozikowski, Alan, Bishai, William
Formato: Artigo
Idioma:Inglês
Publicado em: American Society for Microbiology 2015
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4604386/
https://ncbi.nlm.nih.gov/pubmed/26303802
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.01341-15
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