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Ritonavir is the best alternative to ketoconazole as an index inhibitor of cytochrome P450-3A in drug–drug interaction studies

AIMS: The regulatory prohibition of ketoconazole as a CYP3A index inhibitor in drug–drug interaction (DDI) studies has compelled consideration of alternative inhibitors. METHODS: The biomedical literature was searched to identify DDI studies in which oral midazolam (MDZ) was the victim, and the inhi...

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Pubblicato in:Br J Clin Pharmacol
Autori principali: Greenblatt, David J, Harmatz, Jerold S
Natura: Artigo
Lingua:Inglês
Pubblicazione: John Wiley & Sons, Ltd 2015
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4574820/
https://ncbi.nlm.nih.gov/pubmed/25923589
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/bcp.12668
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