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The soluble Y115E–Y117E variant of human glutaminyl cyclase is a valid target for X-ray and NMR screening of inhibitors against Alzheimer disease

Recent developments in molecular pathology and genetics have allowed the identification of human glutaminyl cyclase (hQC) among the abnormal proteins involved in many neurodegenerative disorders. Difficulties in obtaining large quantities of pure protein may limit the use of crystallographic screeni...

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Publicado en:Acta Crystallogr F Struct Biol Commun
Autores principales: DiPisa, Flavio, Pozzi, Cecilia, Benvenuti, Manuela, Andreini, Matteo, Marconi, Guido, Mangani, Stefano
Formato: Artigo
Lenguaje:Inglês
Publicado: International Union of Crystallography 2015
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC4528929/
https://ncbi.nlm.nih.gov/pubmed/26249687
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1107/S2053230X15010389
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