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Brain Penetration and Efficacy of Different Mebendazole Polymorphs in a Mouse Brain Tumor Model

PURPOSE: Mebendazole (MBZ), first used as an antiparasitic drug, shows preclinical efficacy in models of glioblastoma and medulloblastoma. Three different MBZ polymorphs (A, B and C) exist and a detailed assessment of the brain penetration, pharmacokinetics and anti-tumor properties of each individu...

Täydet tiedot

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Bibliografiset tiedot
Julkaisussa:Clin Cancer Res
Päätekijät: Bai, Ren-Yuan, Staedtke, Verena, Wanjiku, Teresia, Rudek, Michelle A, Joshi, Avadhut, Gallia, Gary L., Riggins, Gregory J.
Aineistotyyppi: Artigo
Kieli:Inglês
Julkaistu: 2015
Aiheet:
Linkit:https://ncbi.nlm.nih.gov/pmc/articles/PMC4526400/
https://ncbi.nlm.nih.gov/pubmed/25862759
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1158/1078-0432.CCR-14-2681
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