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Is Ring Breaking Feasible in Relative Binding Free Energy Calculations?

Our interest is relative binding free energy (RBFE) calculations based on molecular simulations. These are promising tools for lead optimization in drug discovery, computing changes in binding free energy due to modifications of a lead compound. However, in the “alchemical” framework for RBFE calcul...

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Dades bibliogràfiques
Publicat a:J Chem Inf Model
Autors principals: Liu, Shuai, Wang, Lingle, Mobley, David L.
Format: Artigo
Idioma:Inglês
Publicat: 2015
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4489933/
https://ncbi.nlm.nih.gov/pubmed/25835054
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jcim.5b00057
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