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Synthesis and evaluation of [(11)C]PBD150, a radiolabeled glutaminyl cyclase inhibitor for the potential detection of Alzheimer’s disease prior to amyloid β aggregation

The phenol of 1-(3-(1H-imidazol-1-yl)propyl)-3-(4-hydroxy-3-methoxyphenyl)thiourea was selectively carbon-11 labelled to generate [(11)C]PBD150 in 7.3% yield from [(11)C]methyl triflate (non-decay corrected; radiochemical purity ≥95%, specific activity = 5.7 Ci/µmol, n=5). Evaluation of [(11)C]PBD15...

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書目詳細資料
發表在:Medchemcomm
Main Authors: Brooks, Allen F., Jackson, Isaac M., Shao, Xia, Kropog, George W., Sherman, Phillip, Quesada, Carole A., Scott, Peter J.H.
格式: Artigo
語言:Inglês
出版: 2015
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在線閱讀:https://ncbi.nlm.nih.gov/pmc/articles/PMC4474278/
https://ncbi.nlm.nih.gov/pubmed/26101580
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/C5MD00148J
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