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Salmeterol Efficacy and Bias in the Activation and Kinase-Mediated Desensitization of β2-Adrenergic Receptors

Salmeterol is a long-acting β2-adrenergic receptor (β2AR) agonist that is widely used as a bronchodilator for the treatment of persistent asthma and chronic obstructive pulmonary disease in conjunction with steroids. Previous studies demonstrated that salmeterol showed weak efficacy for activation o...

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Detalhes bibliográficos
Publicado no:Mol Pharmacol
Main Authors: Gimenez, Luis E., Baameur, Faiza, Vayttaden, Sharat J., Clark, Richard B.
Formato: Artigo
Idioma:Inglês
Publicado em: The American Society for Pharmacology and Experimental Therapeutics 2015
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4429720/
https://ncbi.nlm.nih.gov/pubmed/25784721
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.114.096800
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