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Agonist Activation of a Nicotinic Acetylcholine Receptor

How does an agonist activate a receptor? In this article I consider the activation process in muscle nicotinic acetylcholine receptors (AChRs), a prototype for understanding the energetics of binding and gating in other ligand-gated ion channels. Just as movements that generate gating currents activ...

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Pubblicato in:Neuropharmacology
Autore principale: Auerbach, Anthony
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2014
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4398594/
https://ncbi.nlm.nih.gov/pubmed/25446670
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.neuropharm.2014.10.004
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