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Inhibition of HDAC3 promotes ligand-independent PPARγ activation by protein acetylation

PPARγ (peroxisome proliferator-activated receptor gamma) is a nuclear receptor whose activation is dependent on a ligand. PPARγ activation by exogenous ligands, such as thiazolidinediones (TZDs), is a strategy in the treatment of type 2 diabetes for the improvement of insulin sensitivity. In additio...

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Detalles Bibliográficos
Publicado en:J Mol Endocrinol
Main Authors: Jiang, Xiaoting, Ye, Xin, Guo, Wei, Lu, Hongyun, Gao, Zhanguo
Formato: Artigo
Idioma:Inglês
Publicado: 2014
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC4391273/
https://ncbi.nlm.nih.gov/pubmed/24982244
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1530/JME-14-0066
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