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Reliability and Extension of Quantitative Prediction of CYP3A4-Mediated Drug Interactions Based on Clinical Data

An approach was proposed in 2007 for quantitative predictions of cytochrome P450 (CYP)3A4-mediated drug-drug interactions. It is based on two characteristic parameters: the contribution ratio (CR; i.e., the fraction of victim drug clearance by CYP) and the inhibition ratio (IR) of the inhibitor. Kno...

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Podrobná bibliografie
Vydáno v:AAPS J
Hlavní autoři: Loue, Constance, Tod, Michel
Médium: Artigo
Jazyk:Inglês
Vydáno: Springer US 2014
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC4389753/
https://ncbi.nlm.nih.gov/pubmed/25274605
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1208/s12248-014-9663-y
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