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Artificial human Met agonists based on macrocycle scaffolds

Hepatocyte growth factor (HGF) receptor, also known as Met, is a member of the receptor tyrosine kinase family. The Met–HGF interaction regulates various signalling pathways involving downstream kinases, such as Akt and Erk. Met activation is implicated in wound healing of tissues via multiple biolo...

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Detalhes bibliográficos
Publicado no:Nat Commun
Main Authors: Ito, Kenichiro, Sakai, Katsuya, Suzuki, Yoshinori, Ozawa, Naoya, Hatta, Tomohisa, Natsume, Tohru, Matsumoto, Kunio, Suga, Hiroaki
Formato: Artigo
Idioma:Inglês
Publicado em: Nature Pub. Group 2015
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4382702/
https://ncbi.nlm.nih.gov/pubmed/25758345
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/ncomms7373
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