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A Novel GTP-Binding Inhibitor, FX2149, Attenuates LRRK2 Toxicity in Parkinson’s Disease Models

Leucine-rich repeat kinase-2 (LRRK2), a cytoplasmic protein containing both GTP binding and kinase activities, has emerged as a highly promising drug target for Parkinson’s disease (PD). The majority of PD-linked mutations in LRRK2 dysregulate its GTP binding and kinase activities, which may contrib...

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Vydáno v:PLoS One
Hlavní autoři: Li, Tianxia, He, Xinhua, Thomas, Joseph M., Yang, Dejun, Zhong, Shijun, Xue, Fengtian, Smith, Wanli W.
Médium: Artigo
Jazyk:Inglês
Vydáno: Public Library of Science 2015
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC4376719/
https://ncbi.nlm.nih.gov/pubmed/25816252
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0122461
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