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Transport proteins determine drug sensitivity and resistance in a protozoan parasite, Trypanosoma brucei

Drug resistance in pathogenic protozoa is very often caused by changes to the ‘transportome’ of the parasites. In Trypanosoma brucei, several transporters have been implicated in uptake of the main classes of drugs, diamidines and melaminophenyl arsenicals. The resistance mechanism had been thought...

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Detalhes bibliográficos
Publicado no:Front Pharmacol
Main Authors: Munday, Jane C., Settimo, Luca, de Koning, Harry P.
Formato: Artigo
Idioma:Inglês
Publicado em: Frontiers Media S.A. 2015
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4356943/
https://ncbi.nlm.nih.gov/pubmed/25814953
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3389/fphar.2015.00032
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