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A Mutation in the Intracellular Loop III/IV of Mosquito Sodium Channel Synergizes the Effect of Mutations in Helix IIS6 on Pyrethroid Resistance

Activation and inactivation of voltage-gated sodium channels are critical for proper electrical signaling in excitable cells. Pyrethroid insecticides promote activation and inhibit inactivation of sodium channels, resulting in prolonged opening of sodium channels. They preferably bind to the open st...

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Dades bibliogràfiques
Publicat a:Mol Pharmacol
Autors principals: Wang, Lingxin, Nomura, Yoshiko, Du, Yuzhe, Liu, Nannan, Zhorov, Boris S., Dong, Ke
Format: Artigo
Idioma:Inglês
Publicat: The American Society for Pharmacology and Experimental Therapeutics 2015
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4352587/
https://ncbi.nlm.nih.gov/pubmed/25523031
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.114.094730
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