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Optimizing the sequence of anti-EGFR targeted therapy in EGFR-mutant lung cancer

Metastatic EGFR-mutant lung cancers are sensitive to the first- and second- generation EGFR tyrosine kinase inhibitors (TKIs), gefitinib, erlotinib, and afatinib, but resistance develops. Acquired resistance (AR) to gefitinib or erlotinib occurs most commonly (>50%) via the emergence of a second-...

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Bibliografski detalji
Izdano u:Mol Cancer Ther
Glavni autori: Meador, Catherine B., Jin, Hailing, de Stanchina, Elisa, Nebhan, Caroline A., Pirazzoli, Valentina, Wang, Lu, Lu, Pengcheng, Vuong, Huy, Hutchinson, Katherine E., Jia, Peilin, Chen, Xi, Eisenberg, Rosana, Ladanyi, Marc, Politi, Katerina, Zhao, Zhongming, Lovly, Christine M., Cross, Darren A. E., Pao, William
Format: Artigo
Jezik:Inglês
Izdano: 2014
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC4338015/
https://ncbi.nlm.nih.gov/pubmed/25477325
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1158/1535-7163.MCT-14-0723
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