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Cabozantinib Loaded DSPE-PEG(2000) Micelles as Delivery System: Formulation, Characterization and Cytotoxicity Evaluation

Cabozantinib, a potent pan-tyrosine kinase inhibitor, has been reported to provide enhanced antitumor efficacy by simultaneously inhibiting both MET and VEGF pathways, which are critical to tumor angiogenesis, survival and migration. It's very poor water solubility prevents its administration b...

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Библиографические подробности
Опубликовано в: :BAOJ Pharm Sci
Главные авторы: Yang, Qiuhong, Moulder k, Ryan, Cohen, Mark S, Cai, Shuang, Forrest, Laird M
Формат: Artigo
Язык:Inglês
Опубликовано: 2015
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC4327881/
https://ncbi.nlm.nih.gov/pubmed/25688382
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