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Interaction Potential of the Multitargeted Receptor Tyrosine Kinase Inhibitor Dovitinib with Drug Transporters and Drug Metabolising Enzymes Assessed in Vitro

Dovitinib (TKI-258) is under development for the treatment of diverse cancer entities. No published information on its pharmacokinetic drug interaction potential is available. Thus, we assessed its interaction with important drug metabolising enzymes and drug transporters and its efficacy in multidr...

Täydet tiedot

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Bibliografiset tiedot
Julkaisussa:Pharmaceutics
Päätekijät: Weiss, Johanna, Theile, Dirk, Dvorak, Zdenek, Haefeli, Walter Emil
Aineistotyyppi: Artigo
Kieli:Inglês
Julkaistu: MDPI 2014
Aiheet:
Linkit:https://ncbi.nlm.nih.gov/pmc/articles/PMC4279137/
https://ncbi.nlm.nih.gov/pubmed/25521244
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/pharmaceutics6040632
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