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Interaction Potential of Etravirine with Drug Transporters Assessed In Vitro
Etravirine is a novel nonnucleoside reverse transcriptase inhibitor (NNRTI) for the treatment of HIV-1 infections. ABC transporters potentially mediate clinically relevant drug-drug interactions. We assessed substrate characteristics and the inhibitory and inductive potential of etravirine on ABC tr...
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| Autors principals: | , , |
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| Format: | Artigo |
| Idioma: | Inglês |
| Publicat: |
American Society for Microbiology (ASM)
2011
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| Matèries: | |
| Accés en línia: | https://ncbi.nlm.nih.gov/pmc/articles/PMC3067076/ https://ncbi.nlm.nih.gov/pubmed/21189339 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.01527-10 |
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