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Allostery in Ca(2+) channel modulation by calcium binding proteins

Distinguishing between allostery and competition among modulating ligands is challenging for large target molecules. Of practical necessity, inferences are often drawn from in vitro assays on target fragments, but such inferences may belie actual mechanisms. One key example of such ambiguity concern...

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Pubblicato in:Nat Chem Biol
Autori principali: Yang, Philemon S., Ben Johny, Manu, Yue, David T.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2014
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4268785/
https://ncbi.nlm.nih.gov/pubmed/24441587
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/nchembio.1436
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