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Allostery in Ca(2+) channel modulation by calcium binding proteins

Distinguishing between allostery and competition among modulating ligands is challenging for large target molecules. Of practical necessity, inferences are often drawn from in vitro assays on target fragments, but such inferences may belie actual mechanisms. One key example of such ambiguity concern...

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Detalles Bibliográficos
Publicado en:Nat Chem Biol
Main Authors: Yang, Philemon S., Ben Johny, Manu, Yue, David T.
Formato: Artigo
Idioma:Inglês
Publicado: 2014
Assuntos:
Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC4268785/
https://ncbi.nlm.nih.gov/pubmed/24441587
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/nchembio.1436
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