Wird geladen...

Role of Desolvation in Thermodynamics and Kinetics of Ligand Binding to a Kinase

[Image: see text] Computer simulations are used to determine the free energy landscape for the binding of the anticancer drug Dasatinib to its src kinase receptor and show that before settling into a free energy basin the ligand must surmount a free energy barrier. An analysis based on using both th...

Ausführliche Beschreibung

Gespeichert in:
Bibliographische Detailangaben
Veröffentlicht in:J Chem Theory Comput
Hauptverfasser: Mondal, Jagannath, Friesner, Richard A., Berne, B. J.
Format: Artigo
Sprache:Inglês
Veröffentlicht: American Chemical Society 2014
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC4263462/
https://ncbi.nlm.nih.gov/pubmed/25516727
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ct500584n
Tags: Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!