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Potentiation of High Voltage–Activated Calcium Channels by 4-Aminopyridine Depends on Subunit Composition
4-Aminopyridine (4-AP, fampridine) is used clinically to improve neuromuscular function in patients with multiple sclerosis, spinal cord injury, and myasthenia gravis. 4-AP can increase neuromuscular and synaptic transmission by directly stimulating high voltage–activated (HVA) Ca(2+) channels indep...
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| Publicado no: | Mol Pharmacol |
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| Main Authors: | , , , , , |
| Formato: | Artigo |
| Idioma: | Inglês |
| Publicado em: |
The American Society for Pharmacology and Experimental Therapeutics
2014
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| Assuntos: | |
| Acesso em linha: | https://ncbi.nlm.nih.gov/pmc/articles/PMC4244593/ https://ncbi.nlm.nih.gov/pubmed/25267719 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.114.095505 |
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