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Discovery of Antibiotics-derived Polymers for Gene Delivery using Combinatorial Synthesis and Cheminformatics Modeling

We describe the combinatorial synthesis and cheminformatics modeling of aminoglycoside antibiotics-derived polymers for transgene delivery and expression. Fifty-six polymers were synthesized by polymerizing aminoglycosides with diglycidyl ether cross-linkers. Parallel screening resulted in identific...

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Dettagli Bibliografici
Pubblicato in:Biomaterials
Autori principali: Potta, Thrimoorthy, Zhen, Zhuo, Grandhi, Taraka Sai Pavan, Christensen, Matthew D., Ramos, James, Breneman, Curt M., Rege, Kaushal
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2013
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4238925/
https://ncbi.nlm.nih.gov/pubmed/24331709
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.biomaterials.2013.10.069
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