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TARGETING THE ONCOGENIC MUC1-C PROTEIN INHIBITS MUTANT EGFR-MEDIATED SIGNALING AND SURVIVAL IN NON-SMALL CELL LUNG CANCER CELLS

PURPOSE: Non-small cell lung cancers (NSCLC) that express the EGF receptor (EGFR) with activating mutations frequently develop resistance to EGFR kinase inhibitors. The mucin 1 (MUC1) heterodimeric protein is aberrantly overexpressed in NSCLC cells and confers a poor prognosis; however, the function...

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Publicat a:Clin Cancer Res
Autors principals: Kharbanda, Akriti, Rajabi, Hasan, Jin, Caining, Tchaicha, Jeremy, Kikuchi, Eiki, Wong, Kwok-Kin, Kufe, Donald
Format: Artigo
Idioma:Inglês
Publicat: 2014
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4219601/
https://ncbi.nlm.nih.gov/pubmed/25189483
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1158/1078-0432.CCR-13-3168
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