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Synthesis and Quantitative Structure–Activity Relationship of Imidazotetrazine Prodrugs with Activity Independent of O6-Methylguanine-DNA-methyltransferase, DNA Mismatch Repair and p53

The antitumor prodrug Temozolomide is compromised by its dependence for activity on DNA mismatch repair (MMR) and the repair of the chemosensitive DNA lesion, O6-methylguanine (O6-MeG), by O6-methylguanine-DNA-methyltransferase (EC 2.1.1.63, MGMT). Tumor response is also dependent on wild-type p53....

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Detalhes bibliográficos
Publicado no:J Med Chem
Main Authors: Pletsas, Dimitrios, Garelnabi, Elrashied A.E., Li, Li, Phillips, Roger M., Wheelhouse, Richard T.
Formato: Artigo
Idioma:Inglês
Publicado em: 2013
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4219134/
https://ncbi.nlm.nih.gov/pubmed/23895620
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm401121k
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