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Combination of the CCL5-Derived Peptide R4.0 with Different HIV-1 Blockers Reveals Wide Target Compatibility and Synergic Cobinding to CCR5

R4.0, a synthetic CCL5/RANTES-derived peptide, exerts potent anti-HIV-1 activity via its nonactivating interaction with CCR5, the major HIV-1 coreceptor. CCR5 chronic activation may promote undesirable inflammatory effects and enhance viral infection; thus, receptor antagonism is a necessary requisi...

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Detalhes bibliográficos
Main Authors: Secchi, Massimiliano, Vassena, Lia, Morin, Sébastien, Schols, Dominique, Vangelista, Luca
Formato: Artigo
Idioma:Inglês
Publicado em: American Society for Microbiology 2014
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4187945/
https://ncbi.nlm.nih.gov/pubmed/25114130
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.03559-14
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