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NL-103, a novel dual-targeted inhibitor of histone deacetylases and hedgehog pathway, effectively overcomes vismodegib resistance conferred by Smo mutations

Misregulation of hedgehog (Hh) signaling has been implicated in the pathogenesis of basal cell carcinoma (BCC) and medulloblastoma. Vismodegib, an orally bioavailable Hh signal pathway inhibitor targeting Smo, has been approved for the treatment of advanced BCC. However, acquired drug resistance to...

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Главные авторы: Zhao, Jie, Quan, Haitian, Xie, Chengying, Lou, Liguang
Формат: Artigo
Язык:Inglês
Опубликовано: Blackwell Publishing Ltd 2014
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC4186412/
https://ncbi.nlm.nih.gov/pubmed/25505589
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/prp2.43
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