Lanean...

Improving the Serum Stability of Site-Specific Antibody Conjugates with Sulfone Linkers

[Image: see text] Current routes for synthesizing antibody–drug conjugates commonly rely on maleimide linkers to react with cysteine thiols. However, thioether exchange with metabolites and serum proteins can compromise conjugate stability and diminish in vivo efficacy. We report the application of...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Egile Nagusiak: Patterson, James T., Asano, Shigehiro, Li, Xiuling, Rader, Christoph, Barbas, Carlos F.
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: American Chemical Society 2014
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC4140540/
https://ncbi.nlm.nih.gov/pubmed/25099687
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/bc500276m
Etiketak: Etiketa erantsi
Etiketarik gabe, Izan zaitez lehena erregistro honi etiketa jartzen!