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Discovery of a Negative Allosteric Modulator of GABA(B) Receptors

[Image: see text] Initialized from the scaffold of CGP7930, an allosteric agonist of GABA(B) receptors, a series of noncompetitive antagonists were discovered. Among these compounds, compounds 3, 6, and 14 decreased agonist GABA-induced maximal effect of IP3 production in HEK293 cells overexpressing...

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Détails bibliographiques
Auteurs principaux: Chen, Lin-Hai, Sun, Bing, Zhang, Yang, Xu, Tong-Jie, Xia, Zhi-Xiong, Liu, Jian-Feng, Nan, Fa-Jun
Format: Artigo
Langue:Inglês
Publié: American Chemical Society 2014
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC4094264/
https://ncbi.nlm.nih.gov/pubmed/25050158
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ml500162z
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