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Identification and synthesis of N-(thiophen-2-yl) benzamide derivatives as BRAF(V600E) inhibitors

The V600E BRAF kinase mutation, which activates the downstream MAPK signaling pathway, commonly occurs in about 8% of all human malignancies and about 50% of all melanomas. In this study, we employed virtual screening and chemical synthesis to identify a series of N-(thiophen-2-yl) benzamide derivat...

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Détails bibliographiques
Auteurs principaux: Xie, Yunfeng, Chen, Xianjie, Qin, Jie, Kong, Xiangqian, Ye, Fei, Jiang, Yuren, Liu, Hong, Jiang, Hualiang, Marmorstein, Ronen, Luo, Cheng
Format: Artigo
Langue:Inglês
Publié: 2013
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC4026330/
https://ncbi.nlm.nih.gov/pubmed/23489628
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2013.02.072
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