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Strategic Use of Plasma and Microsome Binding To Exploit in Vitro Clearance in Early Drug Discovery

[Image: see text] Apparent intrinsic clearance (CLia) determined from microsomal stability assays is a cornerstone in drug discovery. Categorical bins are routinely applied to this end point to facilitate analysis. However, such bins ignore the interdependent nature of apparent intrinsic microsome c...

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Detalhes bibliográficos
Main Authors: Chang, George, Steyn, Stefanus J., Umland, John P., Scott, Dennis O.
Formato: Artigo
Idioma:Inglês
Publicado em: American Chemical Society 2010
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4007956/
https://ncbi.nlm.nih.gov/pubmed/24900175
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ml900012h
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