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Species-specific vesicular monoamine transporter 2 (VMAT2) expression in mammalian pancreatic beta cells: implications for optimising radioligand-based human beta cell mass (BCM) imaging in animal models

AIMS/HYPOTHESIS: Imaging of beta cell mass (BCM) is a major challenge in diabetes research. The vesicular monoamine transporter 2 (VMAT2) is abundantly expressed in human beta cells. Radiolabelled analogues of tetrabenazine (TBZ; a low-molecular-weight, cell-permeant VMAT2-selective ligand) have bee...

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Detalhes bibliográficos
Main Authors: Schäfer, M. K.-H., Hartwig, N. R., Kalmbach, N., Klietz, M., Anlauf, M., Eiden, L. E., Weihe, E.
Formato: Artigo
Idioma:Inglês
Publicado em: 2013
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3955760/
https://ncbi.nlm.nih.gov/pubmed/23404442
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s00125-013-2847-7
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