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A unitary mechanism of calcium antagonist drug action.

[3H]Nitrendipine binding to drug receptor sites associated with calcium channels is allosterically regulated by a diverse group of calcium channel antagonists. Verapamil, D-600 (methoxyverapamil), tiapamil, lidoflazine, flunarizine, cinnarizine, and prenylamine all reduce [3H]nitrendipine binding af...

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Publicado en:Proc Natl Acad Sci U S A
Autores principales: Murphy, K M, Gould, R J, Largent, B L, Snyder, S H
Formato: Artigo
Lenguaje:Inglês
Publicado: National Academy of Sciences 1983
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Acceso en línea:https://ncbi.nlm.nih.govhttps://pmc.ncbi.nlm.nih.gov/articles/PMC393480/
https://ncbi.nlm.nih.govhttps://pubmed.ncbi.nlm.nih.gov/6572372/
https://ncbi.nlm.nih.govhttps://doi.org/10.1073/pnas.80.3.860
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