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Intratumoral concentrations of imatinib after oral administration in patients with glioblastoma multiforme

BACKGROUND: Imatinib, an orally administered tyrosine kinase inhibitor of PDGF receptor, c-abl and c-kit, is currently in clinical trials to assess its efficacy in malignant gliomas. Although imatinib does not readily penetrate an intact blood-brain barrier (BBB), the extent to which it distributes...

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Dettagli Bibliografici
Autori principali: Holdhoff, Matthias, Supko, Jeffrey G., Gallia, Gary L., Hann, Christine L., Bonekamp, David, Ye, Xiaobu, Cao, Bing, Olivi, Alessandro, Grossman, Stuart A.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2009
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3927643/
https://ncbi.nlm.nih.gov/pubmed/19768386
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s11060-009-0008-0
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