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Strategies for Lead Discovery: Application of Footprint Similarity Targeting HIVgp41

A highly-conserved binding pocket on HIVgp41 is an important target for development of anti-viral inhibitors. Holden et al. (Bioorg. Med. Chem. Lett. 2012) recently reported 7 experimentally-verified leads identified through a computational screen to the gp41 pocket in conjunction with a new DOCK sc...

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Autori principali: Holden, Patrick M., Allen, William J., Gochin, Miriam, Rizzo, Robert C.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2013
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3913180/
https://ncbi.nlm.nih.gov/pubmed/24315195
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2013.10.022
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