Učitavanje...

4-Amino-7-chloroquinolines: probing ligand efficiency provides botulinum neurotoxin serotype A light chain inhibitors with significant antiprotozoal activity

Structurally simplified analogs of dual antimalarial and botulinum neurotoxin serotype A light chain (BoNT/A LC) inhibitor bis-aminoquinoline (1) were prepared. New compounds were designed to improve ligand efficiency while maintaining or exceeding the inhibitory potency of 1. Three of the new compo...

Cijeli opis

Spremljeno u:
Bibliografski detalji
Glavni autori: Opsenica, Igor M., Tot, Mikloš, Gomba, Laura, Nuss, Jonathan E., Sciotti, Richard J., Bavari, Sina, Burnett, James C., Šolaja, Bogdan A.
Format: Artigo
Jezik:Inglês
Izdano: 2013
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC3880596/
https://ncbi.nlm.nih.gov/pubmed/23815186
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm4006077
Oznake: Dodaj oznaku
Bez oznaka, Budi prvi tko označuje ovaj zapis!