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Self-Assembled Lipoplexes of Short Interfering RNA (siRNA) Using Spermine-Based Fatty Acid Amide Guanidines: Effect on Gene Silencing Efficiency
Four guanidine derivatives of N(4), N(9)-diacylated spermine have been designed, synthesized, and characterized. These guanidine-containing cationic lipids bound siRNA and formed nanoparticles. Two cationic lipids with C18 unsaturated chains, N(1),N(12)-diamidino-N(4), N(9)-dioleoylspermine and N(1)...
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| Main Authors: | , |
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| Formato: | Artigo |
| Idioma: | Inglês |
| Publicado em: |
MDPI
2011
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| Assuntos: | |
| Acesso em linha: | https://ncbi.nlm.nih.gov/pmc/articles/PMC3857073/ https://ncbi.nlm.nih.gov/pubmed/24310587 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/pharmaceutics3030406 |
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