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Cholinergic Modulation by Opioid Receptor Ligands: Potential Application to Alzheimer’s Disease

Morphinans have a storied history in medicinal chemistry as pain management drugs but have received attention as modulators of cholinergic signaling for the treatment of Alzheimer’s Disease (AD). Galantamine is a reversible, competitive acetylcholinesterase (AChE) inhibitor and allosteric potentiati...

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Détails bibliographiques
Auteurs principaux: Motel, William C., Coop, Andrew, Cunningham, Christopher W.
Format: Artigo
Langue:Inglês
Publié: 2013
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC3816933/
https://ncbi.nlm.nih.gov/pubmed/22931533
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